SCHEMBL9210780

SCHEMBL9210780

COC(=O)c1ccc(C(O)(Cn2ccnc2)c2ccc(-c3ccncc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
CYP26A1 O43174 5/20 0.47
GAA P10253 2/20 0.46
TBXAS1 P24557 2/20 0.42
NPC1 O15118 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
KDM4E B2RXH2 2/20 0.41
CYP19A1 P11511 1/20 0.40
NAMPT P43490 1/20 0.40
AHR P35869 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199981 0.83 CYP11B1 (0.46) MAPTALDH1A1TSHRKDM4ECYP19A1
SCHEMBL9205541 0.82 CYP11B1 (0.47) CYP19A1
SCHEMBL9202390 0.80 KIF11 (0.53) TBXAS1CYP19A1
SCHEMBL9202987 0.79 CYP11B1 (0.48) TSHRKDM4ECYP19A1
SCHEMBL9202252 0.79 CYP17A1 (0.48) CYP19A1
SCHEMBL9205856 0.78 CYP11B1 (0.52) CYP19A1
SCHEMBL10858842 0.77 HTT (0.47) HTTCYP26A1GAATBXAS1MAPT
SCHEMBL13019478 0.75 HDAC1 (0.58) HTTALDH1A1TSHRKDM4E
SCHEMBL741537 0.75 HDAC1 (0.58) HTTALDH1A1TSHRKDM4E
SCHEMBL10863031 0.75 POLB (0.48) HTTCYP26A1GAATBXAS1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513149-B1 PYRIDYLPHENYL NITROGEN HETEROCYCLE-SUBSTITUTED CARBINOLS AND DERIVATIVES THEREOF WITH ANTI-INFLAMMATORY ACTIVITY DU PONT MERCK PHARMA (US) 1995-12-13 EP disclosed
WO-1991011445-A1 PYRIDYLPHENYL NITROGEN HETEROCYCLE-SUBSTITUTED CARBINOLS AND DERIVATIVES THEREOF WITH ANTI-INFLAMMATORY ACTIVITY THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-08-08 WO disclosed