SCHEMBL9211138

SCHEMBL9211138

Cc1nn(C)c2c1CCc1c-2cnn1C

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.44
CSNK2A1 P68400 1/20 0.44
PLK3 Q9H4B4 1/20 0.44
DRD2 P14416 3/20 0.36
DRD4 P21917 3/20 0.36
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9219786 0.98 PLK1 (0.42) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL9211170 0.77 PLK1 (0.44) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL9535703 0.75 PLK1 (0.61) PLK1CSNK2A1PLK3DRD2DRD4
Hydrochloric Acid SCHEMBL9534437 0.73 PLK1 (0.59) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL9211095 0.72 PLK1 (0.49) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL9215010 0.71 PLK1 (0.41) PLK1CSNK2A1PLK3DRD2DRD4
Hydrochloric Acid SCHEMBL9216167 0.70 PLK1 (0.47) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL23889226 0.70 SETD7 (0.45) DRD2DRD4
SCHEMBL9533936 0.68 PLK1 (0.74) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL22980483 0.67 PLK1 (0.79) PLK1CSNK2A1PLK3DRD2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276833-B1 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMA (US) 1995-02-15 EP claimed
EP-0276833-A2 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP claimed
US-4734430-A Dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US claimed