SCHEMBL9211707

SCHEMBL9211707

CSc1ccc(Br)c(CBr)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 8/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34
MAOA P21397 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
AKR1C3 P42330 3/20 0.33
AKR1C2 P52895 3/20 0.33
NOX1 Q9Y5S8 1/20 0.33
MCL1 Q07820 1/20 0.32
CRHR1 P34998 1/20 0.32
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 3/20 0.32
HTR3E A5X5Y0 2/20 0.32
HTR3B O95264 2/20 0.32
HTR1A P08908 2/20 0.32
HTR1D P28221 2/20 0.32
HTR1B P28222 2/20 0.32
HTR1E P28566 2/20 0.32
HTR1F P30939 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19743884 0.83 ALDH1A1 (0.37) SLC6A4SLC6A2SLC6A3HRH3MCL1
SCHEMBL9013249 0.82 MCL1 (0.35) SLC6A4SLC6A2SLC6A3HRH3AKR1C3
SCHEMBL11732988 0.81 NOX1 (0.33) SLC6A4SLC6A2SLC6A3HRH3NOX1
SCHEMBL17119681 0.78 SLC6A4 (0.33) SLC6A4SLC6A2SLC6A3MAOAAKR1C3
SCHEMBL11727833 0.76 SLC6A4 (0.34) SLC6A4SLC6A2SLC6A3NOX1MCL1
SCHEMBL30667643 0.75 MAPT (0.37) SLC6A4SLC6A2SLC6A3MAOAAKR1C3
SCHEMBL27350708 0.75 MAPT (0.37) SLC6A4SLC6A2SLC6A3MAOAAKR1C3
SCHEMBL23393787 0.73 SLC6A4 (0.33) SLC6A4SLC6A2SLC6A3MAOAAKR1C3
SCHEMBL2293428 0.72 NPC1 (0.31)
SCHEMBL30806439 0.71 TAAR1 (0.39) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652875-A1 (HETERO)-ARYL KETONES DERIVATIVES WITH ANTIBACTERIAL PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1995-05-17 EP disclosed
WO-1994002478-A1 (HETERO)-ARYL KETONES DERIVATIVES WITH ANTIBACTERIAL PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1994-02-03 WO disclosed
US-4001233-A CNS STIMULANTS, MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1977-01-04 US disclosed
US-3957787-A CENTRAL NERVOUS SYSTEM STIMULANTS, MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1976-05-18 US disclosed