SCHEMBL9013249

SCHEMBL9013249

CSc1ccc(Br)c(CO)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.35
SLC6A4 P31645 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
HSD17B10 Q99714 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
HPGD P15428 1/20 0.32
AKR1C3 P42330 3/20 0.32
AKR1C2 P52895 3/20 0.32
NOX1 Q9Y5S8 1/20 0.32
HTT P42858 1/20 0.32
CRHR1 P34998 1/20 0.31
NQO2 P16083 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
HTR3E A5X5Y0 2/20 0.31
HTR3B O95264 2/20 0.31
HTR1A P08908 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24009098 0.84 MCL1 (0.35) MCL1SLC6A4SLC6A2SLC6A3HRH3
SCHEMBL11727833 0.82 SLC6A4 (0.34) MCL1SLC6A4SLC6A2SLC6A3HSD17B10
SCHEMBL9211707 0.82 SLC6A4 (0.34) MCL1SLC6A4SLC6A2SLC6A3HRH3
SCHEMBL19743884 0.82 ALDH1A1 (0.37) MCL1SLC6A4SLC6A2SLC6A3HRH3
SCHEMBL8770897 0.81 MCL1 (0.38) MCL1SLC6A4HSD17B10AKR1C3AKR1C2
SCHEMBL24478368 0.80 RHEB (0.30)
SCHEMBL8773468 0.78 MAPT (0.39) MCL1HSD17B10ALDH1A1HPGDAKR1C3
SCHEMBL4459146 0.78 KLF10 (0.50) MCL1ALDH1A1HTR3EHTR3BHTR1A
SCHEMBL6036667 0.76 MCL1 (0.35) MCL1SLC6A4HSD17B10ALDH1A1POLB
SCHEMBL8773287 0.76 CA2 (0.38) MCL1SLC6A4SLC6A2SLC6A3AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536745-A (Hetero)-aryl ketones derivatives with antibacterial properties SMITHKLINE BEECHAM P.L.C. (GB) 1996-07-16 US disclosed
EP-0652875-A1 (HETERO)-ARYL KETONES DERIVATIVES WITH ANTIBACTERIAL PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1995-05-17 EP disclosed
WO-1994002478-A1 (HETERO)-ARYL KETONES DERIVATIVES WITH ANTIBACTERIAL PROPERTIES SMITHKLINE BEECHAM PLC (GB) 1994-02-03 WO disclosed
US-4001233-A CNS STIMULANTS, MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1977-01-04 US disclosed
US-3957787-A CENTRAL NERVOUS SYSTEM STIMULANTS, MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1976-05-18 US disclosed