SCHEMBL9212427

SCHEMBL9212427

COc1cc2c(cc1OC)CCN(CC1CCN(CCCc3cccnc3)C1)CC2

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.48
ABCG2 Q9UNQ0 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
PTAFR P25105 6/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
HCRTR2 O43614 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9742540 0.93 CHRNB4 (0.49) ABCB1ABCG2CHRM2CHRM1CHRM3
Hydrochloric Acid SCHEMBL9740675 0.92 CHRNB2 (0.45) ABCB1ABCG2PTAFRCHRNB2CHRNB4
SCHEMBL9209351 0.84 CHRNB4 (0.46) ABCB1ABCG2CHRM2CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL9740808 0.83 CHRNB4 (0.45) ABCB1ABCG2CHRM2CHRNB2CHRNB4
SCHEMBL9214021 0.83 CHRNB4 (0.43) ABCB1ABCG2CHRM2CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL9740211 0.82 HRH3 (0.43) CHRM2CHRM1CHRM3
SCHEMBL9215863 0.81 BRD4 (0.40) ABCB1CHRM2CHRM1CHRM3CHRNB2
Hydrochloric Acid SCHEMBL9208814 0.81 CHRNB4 (0.44) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9214611 0.80 PTGER2 (0.48) CHRM2CHRM1CHRM3
SCHEMBL9211758 0.80 PDE4B (0.48) ABCB1CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed