SCHEMBL9211758

SCHEMBL9211758

COc1cc2c(cc1OC)CN(CC1CCN(CCCc3ccncc3)C1)C2

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.48
ABCB1 P08183 5/20 0.46
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
EBP Q15125 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
TMEM97 Q5BJF2 1/20 0.40
HSD11B1 P28845 1/20 0.39
PDE4D Q08499 1/20 0.39
HTR7 P34969 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9204602 0.83 HSD11B1 (0.37) SIGMAR1TMEM97HSD11B1
Hydrochloric Acid SCHEMBL9216937 0.81 SIGMAR1 (0.39) PDE4BSIGMAR1HSD11B1
SCHEMBL9212427 0.80 ABCB1 (0.48) ABCB1CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL9208180 0.79 PDE4B (0.58) PDE4BABCB1PDE4DBCHE
SCHEMBL9210283 0.78 SIGMAR1 (0.42) SIGMAR1HSD11B1
SCHEMBL9212261 0.77 ABCB1 (0.49) ABCB1HTR7DRD3
SCHEMBL9214611 0.77 PTGER2 (0.48) PDE4BBCHE
SCHEMBL9624149 0.75 KDM4E (0.46) PDE4BABCB1EBPSIGMAR1TMEM97
SCHEMBL9217614 0.75 ACHE (0.50) ABCB1HTR7DRD4BCHE
Hydrochloric Acid SCHEMBL10644273 0.74 PDE4B (0.66) PDE4BABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed