SCHEMBL9213161

SCHEMBL9213161

CC1CNCCN1c1cccc(Cl)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 3/20 0.56
HTR3B O95264 3/20 0.56
HTR3A P46098 3/20 0.56
HTR3D Q70Z44 3/20 0.56
HTR3C Q8WXA8 3/20 0.56
ALDH1A1 P00352 1/20 0.56
HTR2C P28335 11/20 0.49
PIM1 P11309 2/20 0.47
PIM3 Q86V86 2/20 0.47
PIM2 Q9P1W9 2/20 0.47
HTR2A P28223 5/20 0.45
HTR2B P41595 4/20 0.45
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
KMT2A Q03164 1/20 0.43
ALOX5 P09917 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29668691 1.00 HTR3E (0.56) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL21098721 0.80 ALOX5 (0.48) HTR2CPIM1PIM3PIM2HTR2A
SCHEMBL21098718 0.80 ALOX5 (0.48) HTR2CPIM1PIM3PIM2HTR2A
SCHEMBL3272320 0.79 HTR2C (0.56) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL17884815 0.79 HTR2C (0.48) HTR2CPIM1PIM3PIM2HTR2A
SCHEMBL30609686 0.79 HTR2C (0.48) HTR2CPIM1PIM3PIM2HTR2A
SCHEMBL3266317 0.79 HTR2C (0.56) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL4885307 0.79 PIM1 (0.47) HTR2CPIM1PIM3PIM2HTR2A
SCHEMBL4881237 0.79 PIM1 (0.47) HTR2CPIM1PIM3PIM2HTR2A
SCHEMBL4881229 0.79 PIM1 (0.47) HTR2CPIM1PIM3PIM2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP disclosed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US disclosed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP disclosed