SCHEMBL9213373

SCHEMBL9213373

CCOC(=O)[C@H](CC)[C@H](Br)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 4/20 0.37
TRPA1 O75762 1/20 0.37
LMNA P02545 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ALOX15 P16050 1/20 0.34
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
SOAT1 P35610 1/20 0.34
PIN1 Q13526 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRM1 P11229 1/20 0.33
AKR1A1 P14550 1/20 0.33
CHRM3 P20309 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9203441 0.87 ALDH1A1 (0.40) ALDH1A1TRPA1LMNAHSD17B10ALOX15
SCHEMBL9285351 0.83 CYP2C19 (0.40) CYP2C19ALDH1A1MGAMGAASI
SCHEMBL9205360 0.83 CYP2C19 (0.40) CYP2C19ALDH1A1MGAMGAASI
SCHEMBL11281019 0.80 CYP2C19 (0.52) CYP2C19ALDH1A1TRPA1LMNAHSD17B10
SCHEMBL4753769 0.80 ALDH1A1 (0.42) CYP2C19ALDH1A1TRPA1LMNAHSD17B10
SCHEMBL4753767 0.80 ALDH1A1 (0.42) CYP2C19ALDH1A1TRPA1LMNAHSD17B10
SCHEMBL15015721 0.80 ALDH1A1 (0.42) CYP2C19ALDH1A1TRPA1LMNAHSD17B10
SCHEMBL30987373 0.80 CYP2C19 (0.50) CYP2C19ALDH1A1TDP1CHRM1AKR1A1
SCHEMBL235849 0.79 ALDH1A1 (0.50) ALDH1A1TRPA1LMNAHSD17B10ALOX15
SCHEMBL3464999 0.75 ALDH1A1 (0.37) CYP2C19ALDH1A1TRPA1LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643710-A1 SYNTHESIS OF OPTICALLY ACTIVE LACTONES FROM L-ASPARTIC ACID AND INTERMEDIATES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-03-22 EP disclosed
US-5322942-A Deprotecting and hydrolyzing protected aspartic acid diester, reacting with nitrosylating agent in presence of hydrogen halide, esterifying, reacting with acyl aryl derivative REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-06-21 US disclosed
WO-1992021675-A1 SYNTHESIS OF OPTICALLY ACTIVE LACTONES FROM L-ASPARTIC ACID AND INTERMEDIATES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1992-12-10 WO disclosed