SCHEMBL9213595

SCHEMBL9213595

CCc1ccc(NS(=O)(=O)c2ccc(-c3cnn4c(O)ncnc34)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.54
KIT P10721 4/20 0.48
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPT P10636 2/20 0.45
TP53 P04637 1/20 0.43
LMNA P02545 1/20 0.43
PTPN2 P17706 2/20 0.43
PTPN1 P18031 2/20 0.43
PTPN5 P54829 2/20 0.43
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 1/20 0.41
NAMPT P43490 1/20 0.41
GHSR Q92847 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214125 0.90 KIT (0.42) UCHL1KITKMT2AMAPTALDH1A1
SCHEMBL9174951 0.89 KIT (0.46) KITKMT2AMAPTLMNAPTPN2
SCHEMBL9167954 0.88 PKM (0.50) UCHL1KITKMT2AMAPTTP53
SCHEMBL9220912 0.88 UQCRB (0.49) UCHL1KITMAPTLMNAPTPN2
SCHEMBL9219528 0.86 CES1 (0.48) KITKMT2AMAPTPTPN2PTPN1
SCHEMBL9169588 0.86 UQCRB (0.46) KMT2AMAPTALDH1A1MEN1
SCHEMBL9216550 0.86 MAPT (0.49) KMT2AMAPTTP53PTPN2PTPN1
SCHEMBL9173978 0.86 UQCRB (0.52) KMT2AMAPTLMNAPTPN5ALDH1A1
SCHEMBL9163477 0.86 KIT (0.48) KITMAPTLMNAALDH1A1GHSR
SCHEMBL9218723 0.86 MAPT (0.49) KMT2AL3MBTL1MAPTTP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269859-B2 Pyrazolotriazine compounds OTSUKA PHARMA CO LTD (JP) 1995-10-18 EP disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed
US-4824834-A TREATING GOUT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-04-25 US disclosed