SCHEMBL9213796

SCHEMBL9213796

COc1ccc2scc(CCN3CCCC(CN4CCc5cc(OC)c(OC)cc5CC4=O)C3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.41
MTNR1B P49286 4/20 0.41
MAPT P10636 2/20 0.40
HCN4 Q9Y3Q4 2/20 0.40
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A4 P31645 1/20 0.37
DRD3 P35462 1/20 0.37
KCNH2 Q12809 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
GAA P10253 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
ABCB1 P08183 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214365 0.95 HCN4 (0.40) MTNR1AMTNR1BMAPTHCN4CYP3A4
SCHEMBL9206494 0.94 MTNR1A (0.41) MTNR1AMTNR1BMAPTHTR1AMEN1
SCHEMBL9205217 0.94 HCN4 (0.40) MAPTHCN4CYP3A4ALOX15CHRM2
SCHEMBL9206867 0.92 MTNR1A (0.39) MTNR1AMTNR1BMAPTHTR1ASLC6A4
SCHEMBL9208988 0.91 HCN4 (0.41) MAPTHCN4CYP3A4ALOX15CHRM2
Hydrochloric Acid SCHEMBL9740138 0.90 CYP3A4 (0.41) MAPTHCN4CYP3A4ALOX15CHRM2
SCHEMBL9210183 0.89 HCN4 (0.40) MAPTHCN4CYP3A4ALOX15CHRM2
SCHEMBL9207815 0.88 HCN4 (0.40) MAPTHCN4CYP3A4ALOX15CHRM2
SCHEMBL9205646 0.88 MEN1 (0.40) MTNR1AMTNR1BMAPTHCN4MEN1
SCHEMBL9217178 0.87 HCN4 (0.39) MAPTHCN4CYP3A4ALOX15CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed