SCHEMBL9214264

SCHEMBL9214264

CCOC(=O)C=C1CCN(C(=O)OC)CC1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
ALDH1A1 P00352 5/20 0.34
ESR2 Q92731 1/20 0.34
LMNA P02545 1/20 0.34
KDM4E B2RXH2 3/20 0.34
PKM P14618 1/20 0.34
POLB P06746 3/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
MAPT P10636 2/20 0.33
ABL1 P00519 1/20 0.33
RIN1 Q13671 1/20 0.33
THRB P10828 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
P2RY12 Q9H244 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214260 1.00 CHRNB2 (0.35) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL18301302 0.93 ALDH1A1 (0.40) ALDH1A1ESR2LMNAKDM4EPOLB
SCHEMBL18301301 0.93 ALDH1A1 (0.40) ALDH1A1ESR2LMNAKDM4EPOLB
SCHEMBL30262299 0.93 ALDH1A1 (0.40) ALDH1A1ESR2LMNAKDM4EPOLB
SCHEMBL18299260 0.88 ESR2 (0.36) ALDH1A1ESR2KDM4EPOLBHTT
SCHEMBL18299258 0.88 ESR2 (0.36) ALDH1A1ESR2KDM4EPOLBHTT
SCHEMBL18044501 0.86 ADORA1 (0.41) ALDH1A1ESR2KDM4EPKMSMN1; SMN2
SCHEMBL18044499 0.86 ADORA1 (0.41) ALDH1A1ESR2KDM4EPKMSMN1; SMN2
SCHEMBL14501401 0.86 ALDH1A1 (0.34) CHRNB2CHRNA4CHRNB4CHRNA3ALDH1A1
SCHEMBL30514890 0.81 CTDSP1 (0.38) ALDH1A1ESR2LMNAKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320032-B1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-01-18 EP disclosed
US-5231184-A Viricide intermediate JANSSEN PHARMACEUTICA N.V. (BE) 1993-07-27 US disclosed
US-5106973-A Viricide intermediates JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-21 US disclosed
US-4992433-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-12 US disclosed
EP-0320032-A1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1989-06-14 EP disclosed