SCHEMBL9215468

SCHEMBL9215468

CCCCc1ccc(Cl)nn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KCNH2 Q12809 1/20 0.39
SLC5A2 P31639 2/20 0.37
NOS2 P35228 1/20 0.35
CYP19A1 P11511 3/20 0.35
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35
CTRC Q99895 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
IDO1 P14902 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL941277 0.94 KCNH2 (0.47) ALDH1A1KCNH2SLC5A2CYP19A1GABRA2
SCHEMBL8551658 0.92 KCNH2 (0.50) ALDH1A1KCNH2SLC5A2CYP19A1GABRA2
SCHEMBL9850641 0.92 KCNH2 (0.50) ALDH1A1KCNH2SLC5A2CYP19A1GABRA2
SCHEMBL3182612 0.87 ALDH1A1 (0.48) ALDH1A1SLC5A2NOS2CYP19A1GABRA2
SCHEMBL19009143 0.82 KCNH2 (0.45) KCNH2SLC5A2NOS2CYP19A1GABRA2
SCHEMBL27602446 0.81 KCNH2 (0.41) KCNH2SLC5A2NOS2CYP19A1GABRA2
SCHEMBL12356537 0.80 KCNH2 (0.59) ALDH1A1KCNH2CYP19A1MIF
SCHEMBL4592210 0.79 ALDH1A1 (0.46) ALDH1A1SLC5A2GAAMAPT
SCHEMBL10843908 0.78 CYP1A2 (0.38) ALDH1A1MEN1KMT2AGAAMAPT
SCHEMBL10843918 0.78 CYP1A2 (0.38) ALDH1A1MEN1KMT2AGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320032-B1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-01-18 EP disclosed
CN-1021328-C PROCESS FOR PREPARING PYRIDAZINAMINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 1993-06-23 CN disclosed
US-5106973-A Viricide intermediates JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-21 US disclosed
US-4992433-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-12 US disclosed
EP-0320032-A1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1989-06-14 EP disclosed
CN-1033274-A The preparation method of new Pyridazinyl amine derivative JANSSEN PHARMACEUTICA NV (BE) 1989-06-07 CN disclosed