SCHEMBL9215503

SCHEMBL9215503

CCc1ncnc(NC(CC)c2ccc(O)cc2)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.47
RPS6KB1 P23443 4/20 0.39
AKT1 P31749 2/20 0.37
ESR1 P03372 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
PGR P06401 1/20 0.36
CHRM2 P08172 1/20 0.36
CYP3A4 P08684 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
AR P10275 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CHRM1 P11229 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
DRD1 P21728 1/20 0.36
TBXA2R P21731 1/20 0.36
PTGS1 P23219 1/20 0.36
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523092 0.99 EGFR (0.46) EGFRRPS6KB1AKT1ESR1LMNA
SCHEMBL8303141 0.86 EGFR (0.38) EGFRRPS6KB1AKT1LMNACRHR1
SCHEMBL9837138 0.85 EGFR (0.47) EGFRRPS6KB1AKT1ESR1LMNA
SCHEMBL9869764 0.84 CRHR1 (0.36) EGFRCRHR1
SCHEMBL9524967 0.83 CRHR1 (0.36) EGFRCRHR1
SCHEMBL9523756 0.82 CRHR1 (0.39) EGFRRPS6KB1AKT1CRHR1
SCHEMBL9193841 0.82 CRHR1 (0.39) EGFRRPS6KB1AKT1MAPTCRHR1
SCHEMBL9526898 0.81 RPS6KB1 (0.39) EGFRRPS6KB1AKT1MAPT
SCHEMBL9084666 0.81 PTGER4 (0.40) EGFRRPS6KB1CRHR1
SCHEMBL9216328 0.81 AURKA (0.42) EGFRRPS6KB1AKT1CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3246281-A None JP disclosed
EP-0370704-B1 Aralkylamine derivatives, preparation thereof and fungicides containing the same UBE INDUSTRIES (JP) 1995-02-01 EP disclosed
EP-0264217-B1 ARALKYLAMINOPYRIMIDINE DERIVATIVE, PROCESS FOR PRODUCING THEREOF AND INSECTICIDE, ACARICIDE AND FUNGICIDE CONTAINING SAID DERIVATIVE AS ACTIVE INGREDIENT UBE INDUSTRIES, LTD. (JP) 1993-06-30 EP disclosed
US-5141941-A ARALKYLAMINE DERIVATIVES, AND FUNGICIDES CONTAINING THE SAME UBE INDUSTRIES, LTD. (JP) 1992-08-25 US disclosed
JP-H03246281-A ARALKYLAMINE DERIVATIVE, ITS PRODUCTION AND FUNGICIDE UBE IND LTD 1991-11-01 JP disclosed
EP-0432894-A1 Fungicidal composition UBE INDUSTRIES, LTD. (JP) 1991-06-19 EP disclosed
EP-0424125-A2 Aralkylamine derivatives, preparation method thereof and fungicides containing the same UBE INDUSTRIES, LTD. (JP) 1991-04-24 EP disclosed
US-4985426-A AGRICULTURAL USE UBE INDUSTRIES, LTD. (JP) 1991-01-15 US disclosed
EP-0370704-A2 Aralkylamine derivatives, preparation thereof and fungicides containing the same UBE INDUSTRIES, LTD. (JP) 1990-05-30 EP disclosed
US-4895849-A Aralkylaminopyrimidine compounds which are useful as for producing thereof and insecticides UBE INDUSTRIES, LTD. (JP) 1990-01-23 US disclosed
EP-0264217-A2 Aralkylaminopyrimidine derivative, process for producing thereof and insecticide, acaricide and fungicide containing said derivative as active ingredient UBE INDUSTRIES, LTD. (JP) 1988-04-20 EP disclosed