SCHEMBL9216101

SCHEMBL9216101

COc1ccc(C(Br)CC(C)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.49
KMT2A Q03164 5/20 0.47
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 3/20 0.47
RAB9A P51151 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
GSK3B P49841 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
FFAR1 O14842 2/20 0.45
CYP1A2 P05177 1/20 0.45
LDHA P00338 1/20 0.44
ATM Q13315 1/20 0.44
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
PLA2G1B P04054 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3646915 0.82 CYP1A2 (0.52) KMT2AALDH1A1CYP1A2CES2CES1
SCHEMBL21199897 0.81 AOC3 (0.53) L3MBTL1KMT2AMEN1RAB9ANPSR1
SCHEMBL628797 0.81 LMNA (0.56) L3MBTL1KMT2AALDH1A1MEN1NPSR1
SCHEMBL27553229 0.79 AOC3 (0.56) L3MBTL1KMT2AALDH1A1MAPTFFAR1
SCHEMBL27553231 0.79 AOC3 (0.56) L3MBTL1KMT2AALDH1A1MAPTFFAR1
SCHEMBL4758820 0.79 BRD4 (0.48) KMT2AMEN1LMNAFFAR1CYP1A2
SCHEMBL3647766 0.79 GSK3B (0.42) ALDH1A1GSK3BCYP1A2
SCHEMBL3649808 0.79 HDAC3 (0.44) KMT2AALDH1A1MEN1NPSR1LMNA
SCHEMBL2655629 0.79 CES2 (0.48) KMT2AALDH1A1MEN1LMNAMAPT
SCHEMBL22319291 0.79 CES2 (0.48) KMT2AALDH1A1MEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633886-A1 PHARMACEUTICALLY ACTIVE BICYCLIC-HETEROCYCLIC AMINES PHARMACIA & UPJOHN COMPANY (US) 1995-01-18 EP disclosed