SCHEMBL9216129

SCHEMBL9216129

CC(Cl)C1=NCCc2sccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.51
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
PIM1 P11309 1/20 0.33
PDGFRA P16234 1/20 0.33
PRKACA P17612 1/20 0.33
LTK P29376 1/20 0.33
GRK5 P34947 1/20 0.33
KDR P35968 1/20 0.33
MAP2K2 P36507 1/20 0.33
FLT3 P36888 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK9 P45984 1/20 0.33
CSNK1A1 P48729 1/20 0.33
CDK8 P49336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867650 0.92 NOS2 (0.45) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL8060969 0.68 NOS2 (1.00) NOS2PLK4CHEK1AURKADAPK3
Iodide SCHEMBL8099764 0.67 NOS2 (0.96) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL12158615 0.64 NOS2 (0.50) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL22995934 0.64 NOS2 (0.59) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL13070848 0.64 NOS2 (0.55) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL17807492 0.63 NOS2 (0.53) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL15267114 0.62 NOS2 (0.47) NOS2PLK4CHEK1AURKADAPK3
SCHEMBL17807494 0.61 NOS2 (0.50) NOS2MAP2K1MAP4K2
SCHEMBL31344191 0.58 NOS2 (0.46) NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0333427-B1 Heterocyclic derivatives SMITHKLINE BEECHAM FARMA (IT) 1995-08-23 EP claimed