SCHEMBL9216635

SCHEMBL9216635

N#CN=C(NCc1cccs1)c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 4/20 0.42
HSD17B10 Q99714 2/20 0.42
HPGD P15428 5/20 0.41
POLB P06746 4/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ESR1 P03372 1/20 0.40
STAT3 P40763 1/20 0.40
ESR2 Q92731 1/20 0.40
USP2 O75604 1/20 0.39
CTNNB1 P35222 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209309 0.76 SMN1; SMN2 (0.43) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL9213875 0.76 KDM4E (0.46) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL9216629 0.76 NPC1 (0.43) NPC1RAB9APOLBSMN1; SMN2ESR1
SCHEMBL9216624 0.76 NPC1 (0.43) NPC1RAB9APOLBSMN1; SMN2ESR1
SCHEMBL16598147 0.76 HPGD (0.61) NPC1RAB9AKDM4EALDH1A1HSD17B10
SCHEMBL9217886 0.76 TLR7 (0.44) ALDH1A1SMN1; SMN2GAA
SCHEMBL7959200 0.74 ALDH1A1 (0.50) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL9216882 0.74 RAB9A (0.39) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL7959203 0.74 ALDH1A1 (0.50) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL9215336 0.70 NPC1 (0.53) NPC1RAB9AKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP claimed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US claimed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP claimed
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP disclosed
US-5272164-A Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1993-12-21 US disclosed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US disclosed
US-5166347-A Hypotensive agents, cardiovascular disorders, antiischemic agents and anticoagulants KIRIN BEER KABUSHIKI KAISHA (JP) 1992-11-24 US disclosed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP disclosed