SCHEMBL9217376

SCHEMBL9217376

Cc1nc2cc3c4c(cccc4c2[nH]1)C(=O)N(CCCCNCCCN1C(=O)c2cccc4c2c(cc2nc(C)[nH]c24)C1=O)C3=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 3/20 0.53
HEXA P06865 4/20 0.46
HEXB P07686 4/20 0.46
OGA O60502 1/20 0.46
MEN1 O00255 1/20 0.45
RGS12 O14924 1/20 0.45
USP2 O75604 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
ATM Q13315 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TLR9 Q9NR96 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
DYRK3 O43781 1/20 0.45
RPS6KB1 P23443 1/20 0.45
EPHA2 P29317 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9050186 0.96 SIRT1 (0.49) SIRT1HEXAHEXBOGAMEN1
SCHEMBL9080071 0.87 FTO (0.54) SIRT1HEXAHEXBOGAMEN1
SCHEMBL9212321 0.80 SIRT1 (0.54) SIRT1HEXAHEXBOGAMEN1
SCHEMBL7709787 0.79 KMT2A (0.46) MEN1USP2POLBMAPTHTT
SCHEMBL9219088 0.77 SIRT1 (0.53) SIRT1HEXAHEXBOGAMEN1
SCHEMBL9042793 0.77 SIRT1 (0.50) SIRT1HEXAHEXBOGAMEN1
SCHEMBL9080075 0.75 SIRT1 (0.59) SIRT1HEXAHEXBOGA
SCHEMBL9079634 0.75 SIRT1 (0.50) SIRT1HEXAHEXBOGAMEN1
SCHEMBL9079400 0.74 SIRT1 (0.52) SIRT1HEXAHEXBOGAMEN1
SCHEMBL9079725 0.74 SIRT1 (0.52) SIRT1HEXAHEXBOGAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995000490-A1 BIS-IMIDE POLYCYCLIC AND HETEROCYCLIC CHROMOPHORES USEFUL AS TUMORICIDALS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-01-05 WO disclosed