SCHEMBL9218409

SCHEMBL9218409

COc1n[c]c2ccccc2c1OC

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 1/20 0.45
KDM4E B2RXH2 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MAPK1 P28482 1/20 0.45
POLB P06746 1/20 0.41
MAPT P10636 3/20 0.34
CASP1 P29466 1/20 0.34
IDO1 P14902 2/20 0.32
SQOR Q9Y6N5 2/20 0.32
EP300 Q09472 1/20 0.32
KAT8 Q9H7Z6 1/20 0.32
BTK Q06187 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL638668 0.81 ALDH1A1 (0.45) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL637848 0.80 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL638669 0.80 KDM4E (0.43) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL637849 0.80 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL7111069 0.75 ALDH1A1 (0.39) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL7447549 0.75 MAPT (0.43) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL2259297 0.71 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP2C19KDM4ESMN1; SMN2
SCHEMBL7107250 0.71 RECQL (0.40) ALDH1A1CYP1A2CYP2C19KDM4EMAPK1
SCHEMBL7110679 0.70 PDPK1 (0.38) ALDH1A1CYP1A2CYP2C19
SCHEMBL7111035 0.70 BRD4 (0.37) ALDH1A1CYP1A2CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP claimed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US claimed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed