SCHEMBL9221122

SCHEMBL9221122

COC(=O)c1cc(OC)ccc1SC(=O)N(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
NR4A2 P43354 1/20 0.43
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PLA2G2A P14555 3/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13159061 0.84 CYP46A1 (0.44) KDM4ENR4A2CA1CA2GAA
SCHEMBL20803216 0.82 ALDH1A1 (0.36) KDM4ECA1CA2GLAGAA
SCHEMBL9857862 0.82 KDM4E (0.40) KDM4ECYP1A2CYP2C19CYP2D6HSD17B10
SCHEMBL2467212 0.82 NR4A2 (0.43) KDM4ENR4A2GAAHSD17B10ALDH1A1
SCHEMBL13159056 0.82 ABL1 (0.49) KDM4ENR4A2PLA2G2AALDH1A1MAPT
SCHEMBL31363552 0.82 ALDH1A1 (0.36) KDM4ECA1CA2GLAGAA
SCHEMBL11165984 0.81 ALDH1A1 (0.43) KDM4ECA1CA2GAAHSD17B10
SCHEMBL2470933 0.81 EGFR (0.48) KDM4ECYP2D6ALDH1A1MAPTPKM
SCHEMBL3483627 0.79 ALDH1A1 (0.40) KDM4EALDH1A1MAPTHTTKMT2A
SCHEMBL3484162 0.79 CPS1 (0.43) GAAALDH1A1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0565721-B1 1,4-BENZOTHIAZEPINE DERIVATIVE KANEKO NOBORU (JP) 1995-07-26 EP disclosed
US-5416066-A FOR THE PREVENTION OF MYOCARDIAL INFARCTION OR INHIBITING MYOCARDIAL NECROSIS KIRIN BREWERY CO., LTD. (JP) 1995-05-16 US disclosed
EP-0565721-A1 1,4-BENZOTHIAZEPINE DERIVATIVE KANEKO, Noboru (JP) 1993-10-20 EP disclosed