SCHEMBL9224893

SCHEMBL9224893

c1ccc2c(c1)Cc1cc(CNC3CCCCCC3)ccc1-2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.51
HTT P42858 1/20 0.47
POLB P06746 2/20 0.46
ALDH1A1 P00352 2/20 0.46
GRIN2B Q13224 1/20 0.45
TSHR P16473 2/20 0.45
ATM Q13315 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CHEK1 O14757 1/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNH2 Q12809 1/20 0.43
HDAC1 Q13547 1/20 0.43
CXCR4 P61073 1/20 0.43
CYP17A1 P05093 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9221031 0.85 HRH3 (0.61) HRH3POLBALDH1A1TSHRRAB9A
SCHEMBL9220147 0.79 EPHX2 (0.59) HTTPOLBALDH1A1RAB9ANPC1
SCHEMBL17674317 0.78 HTT (0.50) HTTALDH1A1TSHRATMNPSR1
SCHEMBL6255707 0.78 KDM4E (0.56) HRH3HTTALDH1A1KMT2A
SCHEMBL22462125 0.76 HTT (0.51) HTTALDH1A1TSHRATMNPSR1
SCHEMBL30289817 0.76 HTT (0.51) HTTALDH1A1TSHRATMNPSR1
SCHEMBL1700604 0.75 TSHR (0.55) HTTALDH1A1TSHRATMNPSR1
SCHEMBL7342269 0.75 ALDH1A1 (0.51) HTTALDH1A1TSHRATMNPSR1
SCHEMBL6483838 0.75 CYP1A2 (0.53) ALDH1A1TSHRRAB9ANPC1TP53
SCHEMBL6482657 0.75 CYP1A2 (0.53) ALDH1A1TSHRRAB9ANPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420348-A Enzyme inhibitors YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0447116-B1 Urea derivatives, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMA CO LTD (JP) 1994-12-14 EP disclosed
US-5258405-A Acetyl coenzyme A cholesterol acetyltransferase inhibitors for cardiovascular disorders and atherosclerosis and antilipemic agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1993-11-02 US disclosed
EP-0447116-A1 Urea derivatives, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-09-18 EP disclosed