SCHEMBL9230581

SCHEMBL9230581

COc1ccc(S(=O)(=O)N(CCCN2CCN(c3ccc(F)cc3)CC2)c2ccccc2OC)cc1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 17/20 0.66
HTR2A P28223 13/20 0.66
HTR2C P28335 13/20 0.66
HTR1A P08908 2/20 0.60
MAPT P10636 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9226646 0.96 HTR7 (0.59) HTR7HTR2AHTR2CHTR1A
Oxalic Acid SCHEMBL9234141 0.96 HTR7 (0.63) HTR7HTR2AHTR2CHTR1AMAPT
Oxalic Acid SCHEMBL9232306 0.92 HTR7 (0.57) HTR7HTR2AHTR2CHTR1AMAPT
SCHEMBL9231146 0.84 HTR7 (0.48) HTR7HTR2AHTR2CHTR1AALDH1A1
Oxalic Acid SCHEMBL9232791 0.81 ALDH1A1 (0.47) HTR7HTR2AHTR2CALDH1A1
Oxalic Acid SCHEMBL9232789 0.81 ALDH1A1 (0.47) HTR7HTR2AHTR2CALDH1A1
SCHEMBL9226838 0.81 HTR7 (0.65) HTR7HTR2AHTR2CHTR1AMAPT
Oxalic Acid SCHEMBL9229197 0.79 HTR7 (0.63) HTR7HTR2AHTR2CHTR1AMAPT
SCHEMBL5657065 0.77 ALDH1A1 (0.51) HTR7HTR2AHTR2CHTR1AMAPT
SCHEMBL5658364 0.77 HTR2A (0.58) HTR7HTR2AHTR2CHTR1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed