SCHEMBL9232013

SCHEMBL9232013

CN(C)C1CCN(c2nc(N3CCOCC3)c3ncnc(OCc4ccccc4)c3n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
TSHR P16473 2/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP11B2 P19099 1/20 0.43
MGMT P16455 1/20 0.42
PIK3CD O00329 4/20 0.42
KDM4E B2RXH2 3/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PRMT5 O14744 2/20 0.41
MTOR P42345 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
PDE10A Q9Y233 1/20 0.39
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8851415 0.84 TSHR (0.43) ALDH1A1TSHRPIK3CDKDM4EGLA
SCHEMBL8851226 0.84 TSHR (0.43) ALDH1A1TSHRPIK3CDKDM4EGLA
SCHEMBL9229772 0.83 PIK3CD (0.42) ALDH1A1MAPK1PIK3CDKDM4EGLA
SCHEMBL8851272 0.82 PIK3CD (0.42) ALDH1A1TSHRPIK3CDKDM4EGLA
SCHEMBL9235896 0.82 ADK (0.47) TSHRPIK3CDHRH4
SCHEMBL8851697 0.81 TSHR (0.41) ALDH1A1TSHRPIK3CDKDM4EGLA
SCHEMBL8852171 0.81 PIK3CD (0.42) ALDH1A1TSHRMAPK1HSD17B10PIK3CD
SCHEMBL9232181 0.81 ADK (0.48) TSHRPIK3CD
SCHEMBL8852164 0.80 PIK3CD (0.42) ALDH1A1TSHRMAPK1HSD17B10PIK3CD
SCHEMBL8851255 0.80 TSHR (0.44) ALDH1A1TSHRPIK3CDKDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed