SCHEMBL9232181

SCHEMBL9232181

CN(C)C1CCN(c2nc(N3CCOCC3)c3ncnc(NCCCc4ccccc4)c3n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADK P55263 4/20 0.48
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
ACHE P22303 1/20 0.41
TSHR P16473 1/20 0.40
TMIGD3 P0DMS9 3/20 0.40
ADORA2A P29274 3/20 0.40
ADORA1 P30542 3/20 0.40
ADORA2B P29275 2/20 0.40
PDE5A O76074 1/20 0.39
MCHR1 Q99705 1/20 0.39
PIK3CD O00329 3/20 0.39
HTT P42858 1/20 0.39
KHK P50053 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9235896 0.95 ADK (0.47) ADKPDE4APDE4BPDE4CPDE4D
SCHEMBL9233960 0.82 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9232013 0.81 ALDH1A1 (0.47) TSHRPIK3CD
SCHEMBL8851152 0.80 ADK (0.55) ADKPDE4APDE4BPDE4CPDE4D
SCHEMBL9234793 0.80 KHK (0.44) KHK
SCHEMBL8851226 0.80 TSHR (0.43) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL8851415 0.80 TSHR (0.43) ADKPDE4APDE4BPDE4CPDE4D
SCHEMBL9230367 0.80 PIK3CA (0.46) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL10657965 0.80 KHK (0.51) ADKPDE4APDE4BPDE4CPDE4D
SCHEMBL9229772 0.79 PIK3CD (0.42) PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed