SCHEMBL9234751

SCHEMBL9234751

COc1ccc(CCN(C)c2ncnc3c(N4CCOCC4)nc(Cl)nc23)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
ALOX15 P16050 1/20 0.44
GAK O14976 3/20 0.43
PDE4B Q07343 2/20 0.42
PDE4A P27815 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE11A Q9HCR9 1/20 0.42
PDE10A Q9Y233 2/20 0.39
KDM4E B2RXH2 2/20 0.39
PRKDC P78527 1/20 0.39
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
LRRK2 Q5S007 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10664494 0.88 LMNA (0.45) SMN1; SMN2LMNAKMT2AMEN1KDM4E
SCHEMBL8851087 0.84 MEN1 (0.46) SMN1; SMN2LMNAKMT2AMEN1ALOX15
SCHEMBL8851150 0.81 PDE10A (0.48) SMN1; SMN2LMNAKMT2APDE10AKDM4E
SCHEMBL10657517 0.79 SMN1; SMN2 (0.47) SMN1; SMN2LMNAKMT2AMEN1ALOX15
SCHEMBL8851118 0.78 PDE10A (0.47) KMT2APDE10AKDM4EALDH1A1
SCHEMBL8851490 0.78 SMN1; SMN2 (0.42) SMN1; SMN2LMNAKMT2AMEN1GAK
SCHEMBL8851202 0.78 PDE10A (0.45) SMN1; SMN2LMNAKMT2APDE10AKDM4E
SCHEMBL8851222 0.77 POLB (0.46) SMN1; SMN2LMNAKMT2APDE4BPDE4A
SCHEMBL8851433 0.76 PDE10A (0.48) KMT2APDE4BPDE4APDE4CPDE4D
SCHEMBL10658148 0.74 LMNA (0.42) SMN1; SMN2LMNAKMT2AMEN1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed