SCHEMBL9235804

SCHEMBL9235804

CN([C]=O)c1ccccc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.41
NEK2 P51955 1/20 0.41
LIMK1 P53667 1/20 0.41
DYRK1A Q13627 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
CYP3A4 P08684 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALOX15 P16050 2/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
TDP1 Q9NUW8 3/20 0.34
ALDH1A1 P00352 6/20 0.33
TSHR P16473 5/20 0.33
GAA P10253 4/20 0.33
MAPT P10636 3/20 0.33
HSD17B10 Q99714 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9396470 0.78 CHEK1 (0.41) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL2093822 0.76 TSHR (0.39) CYP3A4SMN1; SMN2ALDH1A1TSHRGAA
SCHEMBL16838887 0.75 CHEK1 (0.45) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL2092838 0.74 ACHE (0.36) SMN1; SMN2TDP1ALDH1A1TSHRGAA
SCHEMBL2089946 0.74 TSHR (0.38) SMN1; SMN2ALDH1A1TSHRGAAMAPT
SCHEMBL2090250 0.74 C1R (0.37) SMN1; SMN2ALDH1A1TSHRGAAMAPT
SCHEMBL10532261 0.74 ALDH1A1 (0.33) SMN1; SMN2ALDH1A1TSHRGAAMAPT
SCHEMBL15268120 0.74 CHEK1 (0.48) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL113870 0.74 CHEK1 (0.60) CHEK1NEK2LIMK1DYRK1ACLK4
SCHEMBL29707613 0.74 CHEK1 (0.60) CHEK1NEK2LIMK1DYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0638553-A1 Carboxylic acid amides having a terminal carboxylic acid group as aggregation inhibiting drugs Dr. Karl Thomae GmbH (DE) 1995-02-15 EP claimed