SCHEMBL9236248

SCHEMBL9236248

Cc1ccc(C[C@@H]2CN(C(=O)CCc3cccnc3)CCN2C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.43
GAA P10253 1/20 0.40
GFER P55789 1/20 0.39
RAB9A P51151 1/20 0.39
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA4 P22748 4/20 0.38
CA9 Q16790 4/20 0.38
C3AR1 Q16581 3/20 0.38
NAMPT P43490 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8475440 1.00 TACR1 (0.43) TACR1GAAGFERRAB9ACA1
SCHEMBL8478209 0.90 TACR1 (0.51) TACR1CA1CA2CA4CA9
SCHEMBL9241594 0.90 TACR1 (0.51) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8480146 0.87 TACR1 (0.43) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL9233966 0.87 TACR1 (0.43) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7556699 0.85 TACR1 (0.42) TACR1
SCHEMBL9235672 0.83 NAMPT (0.44) TACR1NAMPT
SCHEMBL8836563 0.83 NAMPT (0.44) TACR1NAMPT
SCHEMBL9234523 0.83 NAMPT (0.44) TACR1NAMPT
SCHEMBL9235668 0.83 NAMPT (0.44) TACR1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655442-A1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-05-31 EP disclosed