SCHEMBL9237244

SCHEMBL9237244

CCOC(=O)C(C)(C(=O)O)c1ccsc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 1/20 0.40
PIN1 Q13526 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 2/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910119 0.92 CYP1A2 (0.40) MMP8PIN1CYP1A2CYP2C9CYP2C19
SCHEMBL3179603 0.83 CNR2 (0.46) MMP8PIN1CYP1A2CYP2C9CYP2C19
SCHEMBL11367656 0.82 PIN1 (0.37) MMP8PIN1CYP1A2CYP2C9CYP2C19
SCHEMBL10806885 0.82 LCK (0.43) CYP1A2MAPTKMT2AHPGDPPARA
SCHEMBL11082470 0.81 PIN1 (0.38) MMP8PIN1CYP1A2CYP2C9CYP2C19
SCHEMBL11367652 0.80 CYP1A2 (0.39) MMP8PIN1CYP1A2CYP2C9CYP2C19
SCHEMBL2912931 0.79 PIN1 (0.51) MMP8PIN1CYP1A2CYP2C19POLB
SCHEMBL14747879 0.79 PIN1 (0.51) MMP8PIN1CYP1A2CYP2C19POLB
SCHEMBL25308703 0.78 TSHR (0.42) CYP1A2CYP2C9CYP2C19POLBALDH1A1
SCHEMBL9831106 0.77 TSHR (0.39) PIN1CYP1A2CYP2C9CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5418250-A Hypotensive SMITHKLINE BEECHAM CORPORATION (US) 1995-05-23 US disclosed
US-5185351-A Hypotensive agents; for treatment of congestive heart failure, renal failure and glaucoma SMITHKLINE BEECHAM CORPORATION (US) 1993-02-09 US disclosed