SCHEMBL9239604

SCHEMBL9239604

NCCn1ccc2c1-c1ccccc1C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 13/20 0.40
HTR2C P28335 10/20 0.40
MAOA P21397 1/20 0.37
HRH1 P35367 2/20 0.37
PNMT P11086 1/20 0.37
RXRA P19793 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CHRM2 P08172 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
CHRM1 P11229 1/20 0.35
DRD1 P21728 1/20 0.35
SLC6A2 P23975 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8874318 0.88 CYP3A4 (0.41) HTR2AHTR2CMAOAHRH1RXRA
Fumaric Acid SCHEMBL8874309 0.88 CYP3A4 (0.41) HTR2AHTR2CMAOAHRH1RXRA
SCHEMBL7284322 0.87 HTR2A (0.44) HTR2AHTR2CHRH1KDM4ENPC1
SCHEMBL9238629 0.84 CYP2A6 (0.40) HTR2AMAOAMAPTHPGD
SCHEMBL9232942 0.78 KMT2A (0.38) HTR2AHTR2CMAOAHRH1KDM4E
SCHEMBL9239106 0.75 HTR2C (0.69) HTR2AHTR2CKDM4EALDH1A1HPGD
Fumaric Acid SCHEMBL8874359 0.74 MITF (0.40) HTR2AHTR2CMAOAHRH1RXRA
SCHEMBL12758127 0.73 DRD1 (0.46) MAOAKDM4ENPC1ALDH1A1LMNA
SCHEMBL4359389 0.71 HTR2C (0.40) HTR2AHTR2CMAOAHRH1PNMT
SCHEMBL9233567 0.70 BCHE (0.37) HTR2AHTR2CPNMTADRA2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057083-C Tricyclic 1-aminoethylpyrrol derivative HOFFMANN LA ROCHE (CH) 2000-10-04 CN disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed