SCHEMBL9242016

SCHEMBL9242016

COc1ccc(Cn2c(N)nc3nc[nH]c3c2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.56
NPC1 O15118 1/20 0.54
PNP P00491 2/20 0.54
OPRK1 P41145 1/20 0.48
PDE4A P27815 2/20 0.47
PDE4B Q07343 2/20 0.47
PDE4C Q08493 2/20 0.47
PDE4D Q08499 2/20 0.47
MAPT P10636 2/20 0.47
PDE5A O76074 1/20 0.46
TYMS P04818 1/20 0.44
ADORA3 P0DMS8 2/20 0.44
ADORA2B P29275 1/20 0.44
TLR7 Q9NYK1 2/20 0.43
PIN1 Q13526 1/20 0.42
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
BRD4 O60885 1/20 0.41
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3303816 0.86 KDM4E (0.51) KDM4ENPC1PNPPDE4APDE4B
SCHEMBL17186441 0.86 ADORA3 (0.48) KDM4ENPC1PNPOPRK1PDE4A
Hydrochloric Acid SCHEMBL17186519 0.85 ADORA3 (0.47) KDM4ENPC1PNPOPRK1PDE4A
Hydrochloric Acid SCHEMBL18605970 0.85 KDM4E (0.50) KDM4ENPC1PNPPDE4APDE4B
Hydrochloric Acid SCHEMBL17186506 0.85 PNP (0.53) KDM4ENPC1PNPOPRK1PDE4A
SCHEMBL3308563 0.85 PNP (0.51) NPC1PNPPDE4APDE4BPDE4C
SCHEMBL1262627 0.85 PNP (0.51) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL1533551 0.84 MPO (0.54) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL3021043 0.84 PNP (0.50) KDM4EPNPPDE4APDE4BPDE4C
SCHEMBL3310277 0.84 PNP (0.50) PNPPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7278146-A None JP disclosed
CN-100379750-C Inhibitors of nucleoside phosphorylases and nucleosidases EINSTEIN COLL MED (US) 2008-04-09 CN disclosed
CN-1692120-A Nucleoside phosphorylase and nucleosidase inhibitors EINSTEIN COLL MED (US) 2005-11-02 CN disclosed
JP-H07278146-A BENZYLGUANINE DERIVATIVE TOAGOSEI CO LTD 1995-10-24 JP disclosed