SCHEMBL924320

SCHEMBL924320

O=c1oc(-c2ccccc2NS(=O)(=O)c2ccc(F)cc2)nc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 1.00
GAA P10253 1/20 1.00
KMT2A Q03164 4/20 0.84
MEN1 O00255 3/20 0.84
ALDH1A1 P00352 2/20 0.80
LMNA P02545 2/20 0.74
C1R P00736 7/20 0.56
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
F2 P00734 2/20 0.50
PLG P00747 1/20 0.50
KLK1 P06870 1/20 0.50
PRSS1 P07477 1/20 0.50
C1S P09871 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
PTPN2 P17706 2/20 0.49
PTPN1 P18031 2/20 0.49
PTPN5 P54829 2/20 0.49
HSPD1 P10809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5975597 0.92 KMT2A (1.00) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL10819490 0.91 KMT2A (0.88) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL9528544 0.90 KMT2A (0.86) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL5975754 0.89 KMT2A (0.84) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL9528246 0.89 MAPT (1.00) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL9527940 0.86 KMT2A (0.79) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL7185309 0.86 KMT2A (0.79) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL2314299 0.85 KMT2A (1.00) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL30183217 0.85 KMT2A (1.00) MAPTGAAKMT2AMEN1ALDH1A1
SCHEMBL8524818 0.82 MAPT (0.68) MAPTGAAKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180625-B1 MODULATING AND NORMALIZING AN IMPAIRED HAEMOSTATIC BALANCE IN A MAMMAL, WHICH METHOD COMPRISES ADMINISTERING AN EFFECTIVE AMOUNT OF NOVEL BENZOXAZIN DERIVATIVES; ANTICOAGULANTS NOVO NORDISK A/S (DK) 2001-01-30 US claimed
US-7872052-B2 Use of heterocyclic compounds as SCCE inhibitors AREXIS AB (SE) 2011-01-18 US disclosed
US-20060258651-A1 Use of heterocyclic compounds as scce inhibitors QUANTUM LTO HOLDINGS, LLC 2006-11-16 US disclosed
US-6180625-B1 MODULATING AND NORMALIZING AN IMPAIRED HAEMOSTATIC BALANCE IN A MAMMAL, WHICH METHOD COMPRISES ADMINISTERING AN EFFECTIVE AMOUNT OF NOVEL BENZOXAZIN DERIVATIVES; ANTICOAGULANTS NOVO NORDISK A/S (DK) 2001-01-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060258651-A1 Use of heterocyclic compounds as scce inhibitors RCE1, CTSE, SPINT2 MAPT 2054/4885GAA 1036/4885KMT2A 2584/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.