SCHEMBL9244757

SCHEMBL9244757

O=C(O)[C@H]1CC[C@H](c2nnc(-c3ccc(C4CCNCC4)cc3)s2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
CSNK2A2 P19784 1/20 0.40
CSNK2A1 P68400 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2C P18825 1/20 0.40
HRH1 P35367 1/20 0.40
DGAT1 O75907 7/20 0.39
SOAT1 P35610 1/20 0.39
SLC18A3 Q16572 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
P2RY14 Q15391 4/20 0.38
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
TSHR P16473 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9244763 1.00 NPC1 (0.50) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
Hydrochloric Acid SCHEMBL9408018 0.99 NPC1 (0.49) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
Hydrochloric Acid SCHEMBL9407956 0.99 NPC1 (0.49) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
SCHEMBL9407972 0.86 DGAT1 (0.41) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
SCHEMBL9407975 0.86 DGAT1 (0.41) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
Hydrochloric Acid SCHEMBL9408043 0.85 DGAT1 (0.41) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
Hydrochloric Acid SCHEMBL9408112 0.85 DGAT1 (0.41) NPC1RAB9ACSNK2A2CSNK2A1ADRA2A
SCHEMBL9408121 0.84 DGAT1 (0.38) RAB9ADGAT1P2RY14GSK3BDYRK1A
SCHEMBL9408125 0.84 DGAT1 (0.38) RAB9ADGAT1P2RY14GSK3BDYRK1A
SCHEMBL13098792 0.84 NPC1 (0.48) NPC1RAB9ACSNK2A2CSNK2A1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608858-A1 5-Membered heterocycles as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-08-03 EP claimed
JP-7002851-A None JP disclosed
JP-H072851-A FIVE-MEMBERED HETEROCYCLIC COMPOUND, ITS PREPARATION AND PHARMACEUTICAL CONTAINING IT DR KARL THOMAE GMBH 1995-01-06 JP disclosed
EP-0608858-A1 5-Membered heterocycles as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-08-03 EP disclosed