SCHEMBL9407972

SCHEMBL9407972

COC(=O)[C@H]1CC[C@H](c2nnc(-c3ccc(C4CCNCC4)cc3)s2)CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.41
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
CSNK2A2 P19784 1/20 0.37
CSNK2A1 P68400 1/20 0.37
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2C P18825 1/20 0.36
HRH1 P35367 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
P2RY14 Q15391 2/20 0.35
TGFBR1 P36897 1/20 0.35
ACVR1 Q04771 1/20 0.35
USP25 Q9UHP3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9407975 1.00 DGAT1 (0.41) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1
Hydrochloric Acid SCHEMBL9408112 0.99 DGAT1 (0.41) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1
Hydrochloric Acid SCHEMBL9408043 0.99 DGAT1 (0.41) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1
SCHEMBL9408125 0.89 DGAT1 (0.38) DGAT1GSK3BDYRK1AALDH1A1RAB9A
SCHEMBL9408121 0.89 DGAT1 (0.38) DGAT1GSK3BDYRK1AALDH1A1RAB9A
Hydrochloric Acid SCHEMBL9407959 0.88 MAPT (0.38) DGAT1GSK3BDYRK1AALDH1A1RAB9A
Hydrochloric Acid SCHEMBL9408026 0.88 DGAT1 (0.35) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1
SCHEMBL9244763 0.86 NPC1 (0.50) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1
SCHEMBL9244757 0.86 NPC1 (0.50) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1
SCHEMBL9408053 0.86 NR1H4 (0.39) DGAT1GSK3BDYRK1ACSNK2A2CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608858-A1 5-Membered heterocycles as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-08-03 EP claimed
EP-0608858-A1 5-Membered heterocycles as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-08-03 EP disclosed