SCHEMBL9247689

SCHEMBL9247689

C/C=C/CC1CCC(C#Cc2cnc(-c3ccc(F)c(F)c3)nc2)CC1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.34
CHRNA2 Q15822 2/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
NPY5R Q15761 1/20 0.32
KDM1A O60341 1/20 0.32
GRIN2B Q13224 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9246397 0.91 CHRNB2 (0.32) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9247860 0.88 CHRNB2 (0.33) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9246659 0.88 GRM2 (0.38) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9243069 0.86 CHRNB2 (0.33) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9245976 0.85 FFAR1 (0.35) KDM1A
SCHEMBL9243078 0.84 NPY5R (0.34) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9243073 0.84 NPY5R (0.34) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9245762 0.84 PDGFRB (0.32) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9245767 0.84 PDGFRB (0.32) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL9245772 0.84 PDGFRB (0.32) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447657-A Liquid crystal compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-05 US disclosed