SCHEMBL9248237

SCHEMBL9248237

COc1ccccc1C1(O)CCC(c2ccccc2)(c2ccccc2)[C@H]2CN(C(=O)OC(C)(C)C)CC21

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.68
FNTA P49354 2/20 0.42
FNTB P49356 2/20 0.42
MEN1 O00255 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
ALK Q9UM73 1/20 0.41
RORC P51449 7/20 0.40
PDK2 Q15119 1/20 0.39
PDE4B Q07343 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
USP30 Q70CQ3 1/20 0.38
HTR1A P08908 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546697 1.00 TACR1 (0.68) TACR1FNTAFNTBMEN1CYP3A4
SCHEMBL7885109 1.00 TACR1 (0.68) TACR1FNTAFNTBMEN1CYP3A4
SCHEMBL8957032 0.90 TACR1 (0.66) TACR1FNTAFNTBMEN1CYP3A4
SCHEMBL8956775 0.89 TACR1 (0.54) TACR1FNTAFNTBMEN1CYP3A4
SCHEMBL8873936 0.88 TACR1 (0.52) TACR1MEN1KMT2AALKRORC
SCHEMBL8874860 0.88 TACR1 (0.52) TACR1MEN1KMT2AALKRORC
SCHEMBL8956761 0.88 TACR1 (0.52) TACR1TSHRRORCPDK2USP30
SCHEMBL9244693 0.87 TACR1 (0.49) TACR1TSHRRORCUSP30
SCHEMBL8956952 0.87 TACR1 (0.49) TACR1TSHRRORCUSP30
SCHEMBL8545144 0.84 TACR1 (0.48) TACR1FNTAFNTBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463077-A Exhibit substance P antagonist activity RHONE-POULENC RORER S.A. (FR) 1995-10-31 US disclosed