SCHEMBL8956952

SCHEMBL8956952

CC(C)(C)OC(=O)N1C[C@@H]2[C@H](C1)C(c1ccccc1)(c1ccccc1)CC[C@@]2(O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.49
RORC P51449 11/20 0.46
USP30 Q70CQ3 1/20 0.43
TSHR P16473 2/20 0.43
ALOX15 P16050 1/20 0.43
ATM Q13315 1/20 0.43
GPR119 Q8TDV5 1/20 0.43
NAMPT P43490 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9244693 1.00 TACR1 (0.49) TACR1RORCUSP30TSHRALOX15
SCHEMBL8956761 0.89 TACR1 (0.52) TACR1RORCUSP30TSHRALOX15
SCHEMBL9266367 0.88 RORC (0.46) TACR1RORCUSP30TSHRALOX15
SCHEMBL8546697 0.87 TACR1 (0.68) TACR1RORCUSP30TSHR
SCHEMBL7885109 0.87 TACR1 (0.68) TACR1RORCUSP30TSHR
SCHEMBL9248237 0.87 TACR1 (0.68) TACR1RORCUSP30TSHR
SCHEMBL9003029 0.81 USP30 (0.45) TACR1RORCUSP30TSHRALOX15
SCHEMBL9003033 0.81 USP30 (0.45) TACR1RORCUSP30TSHRALOX15
SCHEMBL9262375 0.81 USP30 (0.45) TACR1RORCUSP30TSHRALOX15
SCHEMBL9270074 0.81 USP30 (0.45) TACR1RORCUSP30TSHRALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5484804-A Perhydroisoindole derivatives as antagonists of substance P RHONE-POULENC RORER S.A. (FR) 1996-01-16 US disclosed
US-5463077-A Exhibit substance P antagonist activity RHONE-POULENC RORER S.A. (FR) 1995-10-31 US disclosed