SCHEMBL9249490

SCHEMBL9249490

Cn1c(-c2ccc(C(=N)N)cc2)nc2cc(C(=O)NCCC(=O)O)ccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.56
HDAC8 Q9BY41 3/20 0.56
HDAC6 Q9UBN7 3/20 0.56
HDAC3 O15379 2/20 0.52
HDAC2 Q92769 2/20 0.52
ITGB3 P05106 3/20 0.50
ITGA2B P08514 3/20 0.50
NAMPT P43490 1/20 0.48
F2 P00734 9/20 0.47
PTGER4 P35408 2/20 0.46
SLC22A2 O15244 1/20 0.44
F10 P00742 1/20 0.44
PLG P00747 1/20 0.44
PLAT P00750 1/20 0.44
PROC P04070 1/20 0.44
HPN P05981 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
NQO2 P16083 1/20 0.44
PRSS3 P35030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9249572 0.94 ITGB3 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9252708 0.92 CHEK2 (0.51) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL8863519 0.90 HDAC1 (0.52) HDAC1HDAC8HDAC6HDAC3HDAC2
Hydrochloric Acid SCHEMBL9255053 0.89 HDAC1 (0.51) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9251361 0.89 HDAC6 (0.55) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9255433 0.89 JAK2 (0.50) HDAC1HDAC8HDAC6ITGB3ITGA2B
SCHEMBL9251884 0.88 HDAC1 (0.50) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9247609 0.88 HDAC6 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9255982 0.87 JAK2 (0.52) ITGB3ITGA2BF2PTGER4JAK2
SCHEMBL9249002 0.87 ITGB3 (0.50) HDAC1HDAC8HDAC6HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US claimed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP claimed
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed