SCHEMBL9250170

SCHEMBL9250170

COC(=O)CCc1ccc(-c2ccc(-c3ccc(C(=N)N)cc3)o2)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 13/20 0.61
ALDH1A1 P00352 1/20 0.56
TOP1 P11387 1/20 0.56
HPGD P15428 1/20 0.56
CASP1 P29466 1/20 0.56
CASP7 P55210 1/20 0.56
HSD17B10 Q99714 1/20 0.56
PRMT1 Q99873 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
TOP2A P11388 1/20 0.55
TOP2B Q02880 1/20 0.55
PRSS1 P07477 4/20 0.52
TMPRSS15 P98073 3/20 0.52
F2 P00734 2/20 0.46
F10 P00742 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9254391 0.86 ST14 (0.54) PRSS1F2F10
SCHEMBL9254014 0.86 NQO2 (0.55) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL9258660 0.85 F2 (0.44) NQO2ALDH1A1HPGDHSD17B10PRSS1
SCHEMBL9255174 0.84 NQO2 (0.67) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL9254388 0.83 F2 (0.43) NQO2PRSS1TMPRSS15F2F10
SCHEMBL9253071 0.82 NQO2 (0.56) NQO2PRSS1TMPRSS15F2F10
SCHEMBL9253124 0.81 F2 (0.45) PRSS1TMPRSS15F2F10
Acetic Acid SCHEMBL3506391 0.80 NQO2 (0.82) NQO2ALDH1A1TOP1HPGDCASP1
SCHEMBL9257420 0.79 F2 (0.48) NQO2PRSS1TMPRSS15F2F10
SCHEMBL23566020 0.79 NQO2 (0.79) NQO2ALDH1A1TOP1HPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed