SCHEMBL9250201

SCHEMBL9250201

CS(=O)(=O)c1cc([N+](=O)[O-])cc(O)c1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 5/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
ALDH1A1 P00352 3/20 0.55
ALOX15 P16050 2/20 0.55
PMP22 Q01453 2/20 0.55
KDM4E B2RXH2 1/20 0.55
TTR P02766 1/20 0.55
CYP1A2 P05177 1/20 0.55
MAPT P10636 1/20 0.55
CYP2C9 P11712 1/20 0.55
HPGD P15428 1/20 0.55
ALOX12 P18054 1/20 0.55
MAPK1 P28482 1/20 0.55
RECQL P46063 1/20 0.55
HIF1A Q16665 1/20 0.55
HSD17B10 Q99714 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HTT P42858 2/20 0.49
GALR3 O60755 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28104172 0.86 MEN1 (0.46) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL9603655 0.84 GPR35 (0.59) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL1530296 0.83 MEN1 (0.70) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL9251144 0.80 ERN1 (0.57) MEN1KMT2AALDH1A1KDM4EMAPT
SCHEMBL1530423 0.79 ALDH1A1 (0.55) GPR35ALDH1A1ALOX15PMP22KDM4E
SCHEMBL31738343 0.79 GPR35 (0.55) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL9743157 0.78 GPR35 (0.75) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL12776832 0.74 GPR35 (0.58) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL2441399 0.74 TSHR (0.42) GPR35MEN1KMT2AALDH1A1ALOX15
SCHEMBL69972 0.73 GPR35 (0.69) GPR35MEN1KMT2AALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446194-A Pharmacologically active catechol derivatives ORION-YHTYMA OY (FI) 1995-08-29 US disclosed
US-5283352-A Transferase inhibitor ORION-YHTYMA OY (FI) 1994-02-01 US disclosed
US-5112861-A Inhibitors of catechol-methyl-transferase enzyme, levodopa ORION-YHTYMA OY (FI) 1992-05-12 US disclosed
US-4963590-A ENZYME INHIBITOR FOR TREATING PARKINSON'S DISEASE ALONG WITH DOPA;POTENTIATION ORION-YHTYMA OY (FI) 1990-10-16 US disclosed