SCHEMBL9252873

SCHEMBL9252873

CC(=O)N1CCC(C(=O)c2ccc(N3CCCCC3)cc2N2CCCCC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPT P10636 4/20 0.41
KMT2A Q03164 3/20 0.41
S100B P04271 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LGMN Q99538 1/20 0.40
GFER P55789 2/20 0.40
CASP6 P55212 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9249516 0.82 CYP2C9 (0.47) ALDH1A1MAPTL3MBTL1KDM4ECYP2C19
SCHEMBL9252527 0.80 HSD11B1 (0.53) ALDH1A1MAPTKMT2AL3MBTL1MEN1
SCHEMBL9254041 0.80 HSD11B1 (0.53) ALDH1A1MAPTKMT2AL3MBTL1MEN1
SCHEMBL9255076 0.79 HSD11B1 (0.54) ALDH1A1MAPTKMT2AL3MBTL1MEN1
SCHEMBL19381318 0.75 GFER (0.51) ALDH1A1MAPTKMT2AS100BL3MBTL1
SCHEMBL9377704 0.75 HSD11B1 (0.51) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL9379111 0.75 HSD11B1 (0.54) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL14982136 0.75 ALDH1A1 (0.56) ALDH1A1MAPTKMT2AS100BL3MBTL1
SCHEMBL19381709 0.73 GFER (0.53) ALDH1A1MAPTKMT2AS100BL3MBTL1
SCHEMBL9249523 0.73 ATM (0.39) ALDH1A1L3MBTL1CYP2C19CYP3A4RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed