SCHEMBL9253022

SCHEMBL9253022

CCCCCCCN(CCc1ccc(OCOCCOC)cc1)C(=O)Nc1ccc(OC)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.50
PPARA Q07869 5/20 0.50
PPARD Q03181 3/20 0.50
PLK1 P53350 1/20 0.46
PLK3 Q9H4B4 1/20 0.46
TSHR P16473 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.42
ALDH1A1 P00352 3/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HPGD P15428 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252619 0.92 HDAC1 (0.51) PPARGPPARAPPARDPLK1PLK3
SCHEMBL9261604 0.87 HDAC1 (0.51) PLK1PLK3TSHRMAPTALDH1A1
SCHEMBL9251911 0.85 HDAC1 (0.53) PLK1PLK3TSHRMAPTALDH1A1
SCHEMBL9255485 0.85 PPARG (0.68) PPARGPPARAPPARD
SCHEMBL9253807 0.84 TSHR (0.54) PPARGPPARAPPARDPLK1PLK3
SCHEMBL8923414 0.84 PPARA (0.56) PPARGPPARAPPARDPLK1PLK3
SCHEMBL7075480 0.83 PPARG (0.49) PPARGPPARAPPARDPLK1PLK3
SCHEMBL9577853 0.83 TSHR (0.56) TSHRMAPTALDH1A1GAAHTT
SCHEMBL9259129 0.83 HDAC1 (0.47) PPARGPPARAPPARDTSHRMEN1
SCHEMBL9257655 0.82 TSHR (0.42) PPARGPPARAPPARDPLK1PLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5422373-A An alkoxybenzyl-alkylene-arylurea anticholesterol, antilipemic agents and enzyme inhibitors BURROUGHS WELLCOME CO. (US) 1995-06-06 US disclosed
EP-0550568-A1 ANTI-ATHEROSCLEROTIC ARYL COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1993-07-14 EP disclosed
WO-1992006075-A1 ANTI-ATHEROSCLEROTIC ARYL COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-04-16 WO disclosed