SCHEMBL9253050

SCHEMBL9253050

O=C(c1ccc(N2CCCC2)cc1)C1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.64
NPC1 O15118 2/20 0.64
RAB9A P51151 2/20 0.64
CYP2C19 P33261 1/20 0.61
HTR2A P28223 3/20 0.56
HTR2C P28335 3/20 0.56
HTR2B P41595 3/20 0.56
MAPT P10636 1/20 0.54
HTT P42858 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
TMEM97 Q5BJF2 7/20 0.50
SIGMAR1 Q99720 7/20 0.50
HTR1A P08908 3/20 0.50
HRH2 P25021 3/20 0.50
HRH1 P35367 3/20 0.50
HRH3 Q9Y5N1 3/20 0.50
ADRA2C P18825 2/20 0.50
ENPP2 Q13822 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2848087 0.88 SMN1; SMN2 (0.77) SMN1; SMN2NPC1RAB9ACYP2C19HTR2A
SCHEMBL9256664 0.85 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9ACYP2C19HTR2A
SCHEMBL4063564 0.85 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL14335634 0.85 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9ACYP2C19HTR2A
SCHEMBL5229150 0.80 TMEM97 (0.56) SMN1; SMN2NPC1RAB9ACYP2C19HTR2A
SCHEMBL9256804 0.80 HTR2A (0.81) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL19950156 0.79 MEN1 (0.60) SMN1; SMN2NPC1RAB9ACYP2C19HTR2A
SCHEMBL5237843 0.79 KMT2A (0.54) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL205216 0.79 SMN1; SMN2 (1.00) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL31449815 0.78 SMN1; SMN2 (0.87) SMN1; SMN2NPC1RAB9ACYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed