SCHEMBL9256664

SCHEMBL9256664

O=C(c1ccc(F)cc1)C1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.68
NPC1 O15118 2/20 0.68
RAB9A P51151 2/20 0.68
CYP2C19 P33261 2/20 0.65
HSD11B1 P28845 6/20 0.63
CYP1A2 P05177 2/20 0.58
CYP3A4 P08684 2/20 0.58
CYP2D6 P10635 2/20 0.58
KDM4E B2RXH2 1/20 0.58
HTR2A P28223 1/20 0.58
CYP2C9 P11712 1/20 0.56
HTT P42858 1/20 0.56
LMNA P02545 1/20 0.55
KMT2A Q03164 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2848087 0.91 SMN1; SMN2 (0.77) SMN1; SMN2NPC1RAB9ACYP2C19HSD11B1
SCHEMBL4063564 0.88 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL14335634 0.88 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9ACYP2C19HSD11B1
SCHEMBL9253050 0.85 SMN1; SMN2 (0.64) SMN1; SMN2NPC1RAB9ACYP2C19CYP2D6
SCHEMBL1653094 0.83 HTT (0.69) SMN1; SMN2NPC1RAB9ACYP2C19CYP2D6
SCHEMBL10600330 0.83 HSD11B1 (0.65) SMN1; SMN2CYP2C19HSD11B1KDM4ECYP2C9
SCHEMBL205216 0.82 SMN1; SMN2 (1.00) SMN1; SMN2NPC1RAB9ACYP2C19CYP3A4
SCHEMBL7492647 0.81 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9ACYP2C19CYP3A4
SCHEMBL6208288 0.81 HSD11B1 (0.67) SMN1; SMN2CYP2C19HSD11B1CYP1A2CYP3A4
SCHEMBL5369606 0.81 TPSAB1 (0.69) SMN1; SMN2NPC1RAB9ACYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed