SCHEMBL9253798

SCHEMBL9253798

CC(C)CN1C(=O)[C@H](NC(=O)Nc2cccc(-c3nnn[nH]3)c2)N=C(C(C)C)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 10/20 0.54
CCKAR P32238 2/20 0.49
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302443 0.88 CCKBR (0.55) CCKBRCCKAR
SCHEMBL9260715 0.87 CCKBR (0.58) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9271901 0.87 CCKBR (0.59) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9301212 0.87 CCKBR (0.56) CCKBR
SCHEMBL7547213 0.86 CCKBR (0.60) CCKBRCCKAR
SCHEMBL7547210 0.86 CCKBR (0.60) CCKBRCCKAR
SCHEMBL9003114 0.86 CCKBR (0.50) CCKBRCCKAR
SCHEMBL9540361 0.85 CCKBR (0.54) CCKBRCCKAR
SCHEMBL8542710 0.84 CCKAR (0.59) CCKBRCCKARCYP3A4MAPTTSHR
SCHEMBL9266105 0.84 CCKBR (0.54) CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5451582-A Cholecystokinins and gastrin receptor antagonists MERCK SHARP & DOHME LTD. (GB) 1995-09-19 US claimed
US-5451582-A Cholecystokinins and gastrin receptor antagonists MERCK SHARP & DOHME LTD. (GB) 1995-09-19 US disclosed