SCHEMBL9253988

SCHEMBL9253988

COC(=O)CCCNS(=O)(=O)c1ccc2c(c1)nc(-c1ccc(C(=N)N)cc1)n2C

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
F2 P00734 11/20 0.42
TMPRSS6 Q8IU80 4/20 0.42
PTGER4 P35408 1/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC3 O15379 2/20 0.39
HDAC2 Q92769 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9253361 0.95 CA1 (0.48) ALDH1A1CA12CA1CA2CA9
SCHEMBL9252892 0.91 CA12 (0.48) ALDH1A1CA12CA1CA2CA9
SCHEMBL9248732 0.89 CA1 (0.50) ALDH1A1CA12CA1CA2CA9
SCHEMBL9251086 0.87 CA1 (0.50) ALDH1A1CA12CA1CA2CA9
SCHEMBL9251150 0.84 HDAC1 (0.50) PTGER4HDAC1HDAC8HDAC6HDAC3
SCHEMBL9252002 0.83 CA1 (0.52) ALDH1A1CA12CA1CA2CA9
Hydrochloric Acid SCHEMBL8863892 0.83 HDAC1 (0.49) PTGER4HDAC1HDAC8HDAC6HDAC3
SCHEMBL9253990 0.82 CA1 (0.47) ALDH1A1CA12CA1CA2CA9
SCHEMBL9254928 0.82 HDAC1 (0.47) CA12CA1CA2CA9F2
SCHEMBL9249307 0.82 HDAC1 (0.47) CA12CA1CA2CA9F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed