SCHEMBL9251086

SCHEMBL9251086

Cn1c(-c2ccc(C(=N)N)cc2)nc2cc(S(=O)(=O)NCCC(=O)O)ccc21

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
ALDH1A1 P00352 2/20 0.47
HDAC1 Q13547 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
F2 P00734 10/20 0.45
TMPRSS6 Q8IU80 3/20 0.43
PTGER4 P35408 1/20 0.43
MEN1 O00255 1/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC2 Q92769 1/20 0.42
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252892 0.94 CA12 (0.48) CA1CA2CA12CA9ALDH1A1
SCHEMBL9253361 0.91 CA1 (0.48) CA1CA2CA12CA9ALDH1A1
SCHEMBL9252002 0.90 CA1 (0.52) CA1CA2CA12CA9ALDH1A1
SCHEMBL9253988 0.87 ALDH1A1 (0.48) CA1CA2CA12CA9ALDH1A1
SCHEMBL9248732 0.85 CA1 (0.50) CA1CA2CA12CA9ALDH1A1
SCHEMBL9252896 0.84 MEN1 (0.50) CA1CA2CA12CA9ALDH1A1
SCHEMBL9249490 0.82 HDAC1 (0.56) HDAC1HDAC8HDAC6F2PTGER4
SCHEMBL9249572 0.79 ITGB3 (0.56) HDAC1HDAC8HDAC6F2PTGER4
SCHEMBL9255124 0.78 HDAC1 (0.50) HDAC1HDAC8HDAC6F2PTGER4
SCHEMBL9251773 0.78 HDAC1 (0.50) HDAC1HDAC8HDAC6F2PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed