SCHEMBL9254470

SCHEMBL9254470

COc1ccc([C@H](N)[C@@H](O)C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 1/20 0.50
GRM6 O15303 1/20 0.50
GRM4 Q14833 1/20 0.50
LDHA P00338 1/20 0.47
PTGS2 P35354 3/20 0.46
AKR1C3 P42330 3/20 0.46
AKR1C2 P52895 3/20 0.46
CYP1A2 P05177 3/20 0.46
PTGS1 P23219 2/20 0.46
CDC42 P60953 1/20 0.46
RAC1 P63000 1/20 0.46
TSHR P16473 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
AOC3 Q16853 2/20 0.45
ACP3 P15309 1/20 0.45
PARP1 P09874 1/20 0.44
PARP10 Q53GL7 1/20 0.44
PARP2 Q9UGN5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6046226 0.84 SLC1A3 (0.51) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL6831820 0.84 LDHA (0.49) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL7082950 0.81 LDHA (0.50) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL6478492 0.81 LDHA (0.50) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL30404277 0.81 LDHA (0.50) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL23298286 0.81 LDHA (0.50) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL5281443 0.79 LDHA (0.52) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL7037842 0.79 LDHA (0.52) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL7042339 0.79 LDHA (0.52) GRM8GRM6GRM4LDHAPTGS2
SCHEMBL9257685 0.79 LMNA (0.43) TSHRACHEALDH1A1GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5476954-A Condensing hydroxyl protected taxane derivative with oxazolidine derivative, decyclizing in acid medium, reacting butoxycarbonyl or benzoyl radical with amine, deprotecting, isolating, purifying product RHONE-POULENC RORER S.A. (FR) 1995-12-19 US disclosed