SCHEMBL9254880

SCHEMBL9254880

COC(=O)CCNC(=O)c1ccc2nc(-c3ccc(C(=N)N)cc3)n(C)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.49
BMPR2 Q13873 1/20 0.46
F10 P00742 2/20 0.44
F2 P00734 1/20 0.44
PLG P00747 1/20 0.44
PLAU P00749 1/20 0.44
PRSS1 P07477 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TMPRSS15 P98073 1/20 0.43
HDAC1 Q13547 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACSS2 Q9NR19 5/20 0.42
HDAC3 O15379 2/20 0.41
HDAC2 Q92769 2/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8863519 0.92 HDAC1 (0.52) NPC1RAB9ATMPRSS15HDAC1HDAC8
Hydrochloric Acid SCHEMBL9255053 0.91 HDAC1 (0.51) NPC1RAB9ATMPRSS15HDAC1HDAC8
SCHEMBL9252708 0.90 CHEK2 (0.51) CHEK2BMPR2F10F2PLG
SCHEMBL9255062 0.87 CHEK2 (0.40) CHEK2F10F2PLGPLAU
SCHEMBL9251150 0.87 HDAC1 (0.50) RAB9AHDAC1HDAC8HDAC6MAPT
SCHEMBL9255533 0.86 NPC1 (0.40) CHEK2F2NPC1RAB9ATMPRSS15
Hydrochloric Acid SCHEMBL8863892 0.86 HDAC1 (0.49) RAB9AHDAC1HDAC8HDAC6MAPT
SCHEMBL9249905 0.85 CHEK2 (0.39) CHEK2NPC1RAB9ATMPRSS15HDAC1
SCHEMBL9571166 0.85 HDAC1 (0.40) CHEK2BMPR2F10F2PLG
SCHEMBL9251884 0.85 HDAC1 (0.50) F10F2PLGHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed