SCHEMBL9255533

SCHEMBL9255533

COC(=O)CCNC(=O)c1cc2nc(-c3ccc(C(=N)N)cc3)n(C)c2cc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
BRD4 O60885 1/20 0.40
HDAC1 Q13547 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC3 O15379 2/20 0.39
HDAC2 Q92769 2/20 0.39
CHEK2 O96017 1/20 0.39
TMPRSS15 P98073 1/20 0.39
PRSS12 P56730 3/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PTGER4 P35408 1/20 0.36
F2 P00734 1/20 0.36
KLK1 P06870 1/20 0.36
KLK5 Q9Y337 1/20 0.36
MTOR P42345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252912 0.93 ITGB3 (0.43) BRD4HDAC1HDAC8HDAC6HDAC3
SCHEMBL9252426 0.91 PRSS12 (0.39) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9255062 0.90 CHEK2 (0.40) BRD4HDAC1HDAC8HDAC6HDAC3
SCHEMBL9249905 0.89 CHEK2 (0.39) NPC1RAB9AHDAC1HDAC8HDAC6
SCHEMBL9256882 0.88 CHEK2 (0.38) BRD4HDAC1HDAC8HDAC6HDAC3
SCHEMBL9251414 0.87 CHEK2 (0.38) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9255518 0.86 CHEK2 (0.41) RAB9ABRD4HDAC1HDAC8HDAC6
Acetic Acid SCHEMBL9256132 0.86 CHEK2 (0.39) NPC1RAB9AHDAC1HDAC8HDAC6
SCHEMBL8863519 0.86 HDAC1 (0.52) NPC1RAB9AHDAC1HDAC8HDAC6
SCHEMBL9254880 0.86 CHEK2 (0.49) NPC1RAB9AHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed