SCHEMBL9255556

SCHEMBL9255556

CC(=O)N1CCC(Cc2ccc(N3CCNCC3Cc3ccccc3)cc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 11/20 0.64
SLC6A3 Q01959 11/20 0.64
SLC6A2 P23975 10/20 0.64
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTR2B P41595 1/20 0.49
MAPK14 Q16539 1/20 0.49
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
TACR3 P29371 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2951055 0.79 SLC6A4 (1.00) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL3026559 0.79 CYP2C9 (0.67) CYP2C9CYP2C19HTR2BMAPK14LMNA
SCHEMBL2952322 0.78 SLC6A4 (0.79) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL10445779 0.78 KDM4E (0.46) LMNAGAATACR3
Hydrochloric Acid SCHEMBL9247465 0.77 KDM4E (0.48) LMNAGAATACR3
SCHEMBL6658178 0.76 SLC6A4 (0.81) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL588656 0.76 SLC6A4 (0.81) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL5543652 0.76 SLC6A4 (0.81) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL588544 0.76 SLC6A4 (0.81) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL12089894 0.76 SLC6A4 (0.71) SLC6A4SLC6A3SLC6A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed