SCHEMBL9255567

SCHEMBL9255567

COC(=O)CCc1ccc(-c2nc(-c3ccc(C(C)N)cc3)cn2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.40
AVPR1B P47901 10/20 0.40
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
NPC1 O15118 2/20 0.36
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
RAB9A P51151 1/20 0.36
SYK P43405 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9259613 0.89 HRH3 (0.40) HRH3AVPR1BADRB2ADRB1
SCHEMBL9248373 0.88 FFAR1 (0.40) HRH3AVPR1B
SCHEMBL9251212 0.87 HRH3 (0.42) HRH3AVPR1BNPC1RAB9A
SCHEMBL9248511 0.87 HRH3 (0.42) HRH3AVPR1BNPC1RAB9ASYK
SCHEMBL9257936 0.85 HRH3 (0.39) HRH3AVPR1BNPC1ADRB2ADRB1
SCHEMBL9250844 0.84 HRH3 (0.42) HRH3AVPR1BTP53MAPTNPC1
SCHEMBL9257104 0.83 HRH3 (0.39) HRH3AVPR1BTP53GAAMAPT
SCHEMBL9259034 0.83 NPC1 (0.42) HRH3NPC1RAB9A
SCHEMBL9259602 0.83 HRH3 (0.40) HRH3AVPR1BTP53NPC1RAB9A
SCHEMBL9257434 0.83 NPC1 (0.42) HRH3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed